PEN (rat)
CAS No. 569364-13-2
PEN (rat)( —— )
Catalog No. M30583 CAS No. 569364-13-2
Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
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Biological Information
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Product NamePEN (rat)
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NoteResearch use only, not for human use.
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Brief DescriptionEndogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
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DescriptionEndogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
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In VitroMouse PEN (mPEN) and rat PEN (rPEN) only differ by one residue at the N-terminal end, whereas human PEN (hPEN) is more divergent and has the sequence PEG instead of PEN.PEN binds and activates a GPCR in the brain.
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetGRK (GPCRK)
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number569364-13-2
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Formula Weight2301.62
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Molecular FormulaC102H169N27O33
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Purity>98% (HPLC)
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SolubilityPBS (pH 7.4):1 mg/mL
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SMILES[H]N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](C(C)C)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Gomes et al (2016) Identification of GPR83 as the receptor for the neuroendocrine peptide PEN. Sci.Signal. 9 ra43 PMID:
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